Small-molecule lipid-bilayer anion transporters for biological applications

  • Nathalie Busschaert
  • , Philip A. Gale*
  • *Corresponding author for this work

Research output: Contribution to journalReview articlepeer-review

173 Citations (Scopus)

Abstract

The development of small-molecule lipid-bilayer anion transporters for potential future use in channel replacement therapy for the treatment of diseases caused by dysregulation of anion transport (such as cystic fibrosis), and in treating cancer by perturbing chemical gradients within cells, thus triggering apoptosis, is an area of intense current interest. This Minireview looks at recent developments in the design of small-molecule transmembrane anion transporters and focuses on the progress so far in employing these compounds in biological systems. Into the cell: The development of small-molecule lipid-bilayer anion transporters for potential future use in channel replacement therapy for the treatment of cystic fibrosis, and in treating cancer by perturbing chemical gradients within cells, is currently an area of intense interest. This Minireview looks at recent developments in the design of small-molecule transmembrane anion transporters and focuses on the progress so far in employing these compounds in biological systems.

Original languageEnglish
Pages (from-to)1374-1382
Number of pages9
JournalAngewandte Chemie - International Edition
Volume52
Issue number5
DOIs
Publication statusPublished - 28-Jan-2013
Externally publishedYes

Keywords

  • anions
  • hydrogen bonding
  • ion transport
  • membranes
  • supramolecular chemistry

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