The relevance of K-i calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor

Hannah Wapenaar, Thea van den Bosch, Niek G. J. Leus, Petra E. van der Wouden, Nikolaos Eleftheriadis, Jos Hermans, Gebremedhin Solomon Hailu, Dante Rotili, Antonello Mai, Alexander Domling, Rainer Bischoff, Hidde J. Haisma, Frank J. Dekker*

*Corresponding author voor dit werk

Onderzoeksoutput: ArticleAcademicpeer review

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Biochemistry, Genetics and Molecular Biology

Pharmacology, Toxicology and Pharmaceutical Science

Chemistry

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